Granisetron hydrochloride

CAS No. 107007-99-8

Granisetron hydrochloride ( BRL 43694 )

Catalog No. M10289 CAS No. 107007-99-8

Granisetron Hcl(BRL 43694A) is a serotonin 5-HT3 receptor antagonist used as an antiemetic to treat nausea and vomiting following chemotherapy.

Purity : >98%(HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
25MG 46 In Stock
50MG 67 In Stock
100MG 116 In Stock
200MG 169 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Granisetron hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Granisetron Hcl(BRL 43694A) is a serotonin 5-HT3 receptor antagonist used as an antiemetic to treat nausea and vomiting following chemotherapy.
  • Description
    Granisetron Hcl(BRL 43694A) is a serotonin 5-HT3 receptor antagonist used as an antiemetic to treat nausea and vomiting following chemotherapy. IC50 Value: 17uM (GR reduced 5-HT-evoked contractions)
  • Synonyms
    BRL 43694
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    107007-99-8
  • Formula Weight
    348.87
  • Molecular Formula
    C18H25ClN4O
  • Purity
    >98%(HPLC)
  • Solubility
    Ethanol: 1 mg/mL (2.86 mM); Water: 70 mg/mL (200.64 mM); DMSO: 1 mg/mL (2.86 mM)
  • SMILES
    Cl.CN1N=C(C(=O)NC2CC3CCCC(C2)N3C)C2=CC=CC=C12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Turvill JL, et al. Br J Pharmacol. 2000 Jul;130(5):1031-6.
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